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Mechanisms of resistance to EZH2 inhibitors in diffuse large B-cell  lymphomas. - Abstract - Europe PMC
Mechanisms of resistance to EZH2 inhibitors in diffuse large B-cell lymphomas. - Abstract - Europe PMC

Targeting EZH2 histone methyltransferase activity alleviates experimental  intestinal inflammation | Nature Communications
Targeting EZH2 histone methyltransferase activity alleviates experimental intestinal inflammation | Nature Communications

A covalently bound inhibitor triggers EZH2 degradation through  CHIP‐mediated ubiquitination | The EMBO Journal
A covalently bound inhibitor triggers EZH2 degradation through CHIP‐mediated ubiquitination | The EMBO Journal

Six Years (2012–2018) of Researches on Catalytic EZH2 Inhibitors: The Boom  of the 2‐Pyridone Compounds - Fioravanti - 2018 - The Chemical Record -  Wiley Online Library
Six Years (2012–2018) of Researches on Catalytic EZH2 Inhibitors: The Boom of the 2‐Pyridone Compounds - Fioravanti - 2018 - The Chemical Record - Wiley Online Library

UTX/KDM6A Loss Enhances the Malignant Phenotype of Multiple Myeloma and  Sensitizes Cells to EZH2 inhibition - ScienceDirect
UTX/KDM6A Loss Enhances the Malignant Phenotype of Multiple Myeloma and Sensitizes Cells to EZH2 inhibition - ScienceDirect

GSK126 inhibits cellular EZH2 methyltransferase activity in multiple... |  Download Scientific Diagram
GSK126 inhibits cellular EZH2 methyltransferase activity in multiple... | Download Scientific Diagram

Identification of EZH2 and EZH1 Small Molecule Inhibitors with Selective  Impact on Diffuse Large B Cell Lymphoma Cell Growth - ScienceDirect
Identification of EZH2 and EZH1 Small Molecule Inhibitors with Selective Impact on Diffuse Large B Cell Lymphoma Cell Growth - ScienceDirect

Pharmacological inhibition of EZH2 by GSK126 decreases atherosclerosis by  modulating foam cell formation and monocyte adhesion in apolipoprotein  E‑deficient mice
Pharmacological inhibition of EZH2 by GSK126 decreases atherosclerosis by modulating foam cell formation and monocyte adhesion in apolipoprotein E‑deficient mice

GSK126 | ≥99%(HPLC) | Selleck | Histone Methyltransferase inhibitor
GSK126 | ≥99%(HPLC) | Selleck | Histone Methyltransferase inhibitor

Inhibitors of the Histone Methyltransferases EZH2/1 Induce a Potent  Antiviral State and Suppress Infection by Diverse Viral Pathogens | mBio
Inhibitors of the Histone Methyltransferases EZH2/1 Induce a Potent Antiviral State and Suppress Infection by Diverse Viral Pathogens | mBio

A covalently bound inhibitor triggers EZH2 degradation through  CHIP‐mediated ubiquitination | The EMBO Journal
A covalently bound inhibitor triggers EZH2 degradation through CHIP‐mediated ubiquitination | The EMBO Journal

Epigenetic‐Based Mechanisms of Osteoblast Suppression in Multiple Myeloma  Bone Disease - Adamik - 2019 - JBMR Plus - Wiley Online Library
Epigenetic‐Based Mechanisms of Osteoblast Suppression in Multiple Myeloma Bone Disease - Adamik - 2019 - JBMR Plus - Wiley Online Library

Inhibition of EZH2 transactivation function sensitizes solid tumors to  genotoxic stress | PNAS
Inhibition of EZH2 transactivation function sensitizes solid tumors to genotoxic stress | PNAS

Enhancer of Zeste Homolog 2 Inhibition Stimulates Bone Formation and  Mitigates Bone Loss Caused by Ovariectomy in Skeletally Mature Mice* -  Journal of Biological Chemistry
Enhancer of Zeste Homolog 2 Inhibition Stimulates Bone Formation and Mitigates Bone Loss Caused by Ovariectomy in Skeletally Mature Mice* - Journal of Biological Chemistry

EZH2 - Wikipedia
EZH2 - Wikipedia

Cancers | Free Full-Text | EZH2 Inhibition as New Epigenetic Treatment  Option for Pancreatic Neuroendocrine Neoplasms (PanNENs) | HTML
Cancers | Free Full-Text | EZH2 Inhibition as New Epigenetic Treatment Option for Pancreatic Neuroendocrine Neoplasms (PanNENs) | HTML

GSK126 inhibits proliferation and causes G2/M cell cycle arrest in EZH2...  | Download Scientific Diagram
GSK126 inhibits proliferation and causes G2/M cell cycle arrest in EZH2... | Download Scientific Diagram

Pharmacological inhibition of EZH2 by GSK126 decreases atherosclerosis by  modulating foam cell formation and monocyte adhesion in apolipoprotein  E‑deficient mice
Pharmacological inhibition of EZH2 by GSK126 decreases atherosclerosis by modulating foam cell formation and monocyte adhesion in apolipoprotein E‑deficient mice

GSK126 causes cell growth inhibition via de-repression of tumor... |  Download Scientific Diagram
GSK126 causes cell growth inhibition via de-repression of tumor... | Download Scientific Diagram

Pharmacological inhibition of EZH2 by GSK126 decreases atherosclerosis by  modulating foam cell formation and monocyte adhesion in apolipoprotein  E‑deficient mice
Pharmacological inhibition of EZH2 by GSK126 decreases atherosclerosis by modulating foam cell formation and monocyte adhesion in apolipoprotein E‑deficient mice

Catalytic Inhibitors of EZH2 Fail to Recapitulate the EZH2 Knockdown... |  Download Scientific Diagram
Catalytic Inhibitors of EZH2 Fail to Recapitulate the EZH2 Knockdown... | Download Scientific Diagram

Frontiers | EZH2 Inhibition Interferes With the Activation of Type I  Interferon Signaling Pathway and Ameliorates Lupus Nephritis in NZB/NZW F1  Mice | Immunology
Frontiers | EZH2 Inhibition Interferes With the Activation of Type I Interferon Signaling Pathway and Ameliorates Lupus Nephritis in NZB/NZW F1 Mice | Immunology

Inhibition of EZH2 transactivation function sensitizes solid tumors to  genotoxic stress | PNAS
Inhibition of EZH2 transactivation function sensitizes solid tumors to genotoxic stress | PNAS

Pharmacological inhibition of EZH2 combined with DNA‑damaging agents  interferes with the DNA damage response in MM cells
Pharmacological inhibition of EZH2 combined with DNA‑damaging agents interferes with the DNA damage response in MM cells

EZH2 - Wikipedia
EZH2 - Wikipedia

Diosgenin and GSK126 Produce Synergistic Effects on Epithelial–M | OTT
Diosgenin and GSK126 Produce Synergistic Effects on Epithelial–M | OTT

Identification and characterization of second-generation EZH2 inhibitors  with extended residence times and improved biological activity - Journal of  Biological Chemistry
Identification and characterization of second-generation EZH2 inhibitors with extended residence times and improved biological activity - Journal of Biological Chemistry

GSK-126 Protects CA1 Neurons from H3K27me3-Mediated Apoptosis in Cerebral  Ischemia | SpringerLink
GSK-126 Protects CA1 Neurons from H3K27me3-Mediated Apoptosis in Cerebral Ischemia | SpringerLink